SCHEMBL2854060

SCHEMBL2854060

O=C(NCc1cc(C(F)(F)F)cc(C(F)(F)F)c1)c1cnn(-c2ccccc2)c1C(F)(F)F

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.65
ALDH1A1 P00352 1/20 0.65
CCR1 P32246 9/20 0.61
MAPT P10636 2/20 0.58
POLB P06746 1/20 0.58
SMN1; SMN2 Q16637 1/20 0.58
DDR1 Q08345 1/20 0.58
MAPK11 Q15759 1/20 0.58
MAPK14 Q16539 1/20 0.58
DDR2 Q16832 1/20 0.58
TMEM97 Q5BJF2 1/20 0.58
MAP3K20 Q9NYL2 1/20 0.58
MAP3K2 Q9Y2U5 1/20 0.58
TDP1 Q9NUW8 1/20 0.55
HPGD P15428 1/20 0.55
TACR1 P25103 1/20 0.54
DGAT2 Q96PD7 1/20 0.51
KMT2A Q03164 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2850396 0.94 KDM4E (0.60) KDM4EALDH1A1CCR1MAPTPOLB
SCHEMBL2857071 0.92 CCR1 (0.57) KDM4EALDH1A1CCR1DDR1MAPK11
SCHEMBL2859642 0.91 CCR1 (0.73) KDM4EALDH1A1CCR1MAPTPOLB
SCHEMBL2857923 0.90 CCR1 (0.66) KDM4EALDH1A1CCR1DDR1MAPK11
SCHEMBL2861147 0.90 KDM4E (0.67) KDM4EALDH1A1CCR1MAPTPOLB
SCHEMBL2860213 0.90 KDM4E (0.73) KDM4EALDH1A1CCR1MAPTPOLB
SCHEMBL2855565 0.89 CCR1 (0.66) KDM4EALDH1A1CCR1MAPT
SCHEMBL2854119 0.88 HPGD (0.73) KDM4ECCR1MAPTPOLBSMN1; SMN2
SCHEMBL2850153 0.88 KDM4E (0.63) KDM4EALDH1A1CCR1MAPTPOLB
SCHEMBL2855701 0.86 CCR1 (0.54) KDM4EALDH1A1CCR1DDR1MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed