SCHEMBL28545430

SCHEMBL28545430

CC(=O)CN(c1ccccc1)c1ccc(C)cc1C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CACNA2D1 P54289 1/20 0.43
CACNA1B Q00975 1/20 0.43
CACNB1 Q02641 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
CRHR1 P34998 2/20 0.41
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
LMNA P02545 2/20 0.40
MTNR1A P48039 1/20 0.40
MTNR1B P49286 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
GAA P10253 1/20 0.39
NPC1 O15118 2/20 0.38
MAPT P10636 1/20 0.38
CASP3 P42574 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38
SENP6 Q9GZR1 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22338052 0.79 TP53 (0.44) CACNA2D1CACNA1BCACNB1MEN1KMT2A
SCHEMBL21969930 0.78 KDM4E (0.42) CACNA2D1CACNA1BCACNB1MEN1KMT2A
SCHEMBL374605 0.78 MTNR1A (0.53) CACNA2D1CACNA1BCACNB1MEN1KMT2A
SCHEMBL22485411 0.76 CYP2C19 (0.47) MEN1KMT2ANPC1MAPTPOLB
SCHEMBL3105534 0.76 MTNR1A (0.52) CACNA2D1CACNA1BCACNB1MEN1KMT2A
SCHEMBL21969562 0.75 MEN1 (0.40) CACNA2D1CACNA1BCACNB1MEN1KMT2A
SCHEMBL23758985 0.75 CACNA2D1 (0.37) CACNA2D1CACNA1BCACNB1MEN1KMT2A
SCHEMBL22485571 0.75 PYCR1 (0.43) MEN1KMT2ALMNASMN1; SMN2NPC1
SCHEMBL22485470 0.75 CYP2C19 (0.46) MEN1KMT2ANPC1MAPTTSHR
SCHEMBL22485618 0.74 ESR1 (0.39) MEN1KMT2ASMN1; SMN2GAANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107074885-B Boronic acid derivatives 默克专利股份公司 2020-11-27 CN disclosed