SCHEMBL28545917

SCHEMBL28545917

CC(C)(C)OC(=O)N(C(=O)OC(C)(C)C)c1nccc2ccc(-n3nc(C(=O)O)cc3C(F)(F)F)cc12

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.40
KLKB1 P03952 3/20 0.36
KDM4E B2RXH2 4/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
PTGER1 P34995 5/20 0.33
CNR1 P21554 2/20 0.33
CNR2 P34972 2/20 0.33
MAPT P10636 1/20 0.32
TSHR P16473 1/20 0.32
MAPK1 P28482 1/20 0.32
CASP1 P29466 1/20 0.32
LDHA P00338 3/20 0.32
POLB P06746 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
HSD17B10 Q99714 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18605021 0.88 GAA (0.40) ALDH1A1KLKB1KDM4EGAAMAPT
SCHEMBL30415347 0.88 GAA (0.40) ALDH1A1KLKB1KDM4EGAAMAPT
SCHEMBL18623280 0.86 KLKB1 (0.33) KLKB1
SCHEMBL31067477 0.84 KLKB1 (0.45) KLKB1
SCHEMBL18604759 0.84 KLKB1 (0.45) KLKB1
SCHEMBL18623250 0.81 F10 (0.40) ALDH1A1KLKB1KDM4EGAATSHR
SCHEMBL17064405 0.78 KLKB1 (0.52) ALDH1A1KLKB1KDM4EGAASMN1; SMN2
SCHEMBL18604730 0.76 KDM4E (0.37) ALDH1A1KDM4ETSHRHSD17B10
SCHEMBL3743397 0.73 PDPK1 (0.37) ALDH1A1KDM4EPOLB
SCHEMBL18623251 0.73 ALDH1A1 (0.46) ALDH1A1KDM4EMAPTPOLBL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113307772-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2024-06-28 CN disclosed
CN-113307772-A Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-08-27 CN disclosed
CN-106257976-B Human plasma kallikrein inhibitors 拜奥克里斯特制药公司 2021-02-02 CN disclosed