SCHEMBL28546709

SCHEMBL28546709

Cc1ccc(CN(C)CC(O)c2cccc(Br)c2)c(C)c1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 2/20 0.44
TAAR1 Q96RJ0 1/20 0.43
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
GRIN1 Q05586 1/20 0.36
GRIN2B Q13224 1/20 0.36
AOC3 Q16853 1/20 0.36
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
ALDH1A1 P00352 1/20 0.36
MAPK1 P28482 1/20 0.36
KDM4E B2RXH2 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
SLC6A3 Q01959 1/20 0.34
SLC18A3 Q16572 1/20 0.34
SIGMAR1 Q99720 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30435410 1.00 PYCR1 (0.44) PYCR1TAAR1SLC6A2SLC6A4GRIN1
SCHEMBL30435138 0.89 PYCR1 (0.43) PYCR1TAAR1SLC6A2SLC6A4AOC3
SCHEMBL28555041 0.89 PYCR1 (0.43) PYCR1TAAR1SLC6A2SLC6A4AOC3
SCHEMBL28911320 0.88 PYCR1 (0.40) PYCR1TAAR1AOC3KMT2AMEN1
SCHEMBL30435089 0.88 PYCR1 (0.40) PYCR1TAAR1AOC3KMT2AMEN1
SCHEMBL20404615 0.80 KMT2A (0.56) PYCR1TAAR1SLC6A2SLC6A4KMT2A
SCHEMBL2578168 0.79 PYCR1 (0.45) PYCR1SLC6A2SLC6A4AOC3KMT2A
SCHEMBL28168731 0.78 MEN1 (0.54) PYCR1TAAR1AOC3KMT2AMEN1
SCHEMBL748686 0.75 TAAR1 (0.49) PYCR1TAAR1KMT2AMEN1ALDH1A1
SCHEMBL20374838 0.75 TAAR1 (0.52) PYCR1TAAR1SLC6A2SLC6A4AOC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112679427-B Tetrahydroisoquinoline derivative, preparation method thereof and application thereof in medicines 江苏恒瑞医药股份有限公司 2023-05-12 CN disclosed
CN-112679427-A Tetrahydroisoquinoline derivatives, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-04-20 CN disclosed