SCHEMBL28547149

SCHEMBL28547149

CCCCCc1ccnc(NC(N)=O)n1

nearest known ligand 0.44

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.44
NR3C2 P08235 4/20 0.38
TRPV1 Q8NER1 5/20 0.38
SPHK1 Q9NYA1 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12609268 0.78 KCNH2 (0.53) KCNH2
SCHEMBL17561037 0.77 DNM2 (0.55) KCNH2
SCHEMBL1231970 0.77 KMT2A (0.49) KCNH2
SCHEMBL1231968 0.77 KCNH2 (0.44) KCNH2SPHK1
SCHEMBL1257991 0.75 NR3C2 (0.43) NR3C2SPHK1
SCHEMBL11034761 0.75 KDM4E (0.38) NR3C2
SCHEMBL14340874 0.74 NPC1 (0.41)
SCHEMBL28551461 0.74 KCNH2 (0.47) KCNH2
SCHEMBL1028320 0.73 KCNH3 (0.56) KCNH2
SCHEMBL11565431 0.73 MAP4K4 (0.50) KCNH2SPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112641787-A Combination therapy comprising a B-Raf inhibitor and a second inhibitor 诺华股份有限公司 2021-04-13 CN disclosed