SCHEMBL28547159

SCHEMBL28547159

CCOc1cc2ncc(C#N)c(Nc3ccc(Cl)cc3)c2cc1N

nearest known ligand 0.70

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
STK4 Q13043 5/20 0.70
SRC P12931 6/20 0.70
EGFR P00533 6/20 0.67
ERBB2 P04626 6/20 0.67
MAP2K1 Q02750 3/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2574073 0.89 EGFR (0.85) STK4SRCEGFRERBB2MAP2K1
SCHEMBL20584416 0.89 EGFR (0.71) STK4SRCEGFRERBB2
SCHEMBL31661487 0.89 MAP2K1 (0.73) STK4SRCEGFRERBB2MAP2K1
Hydrochloric Acid SCHEMBL2052299 0.88 EGFR (0.84) STK4SRCEGFRERBB2MAP2K1
SCHEMBL31661555 0.87 STK4 (0.72) STK4SRCEGFRERBB2
SCHEMBL14135437 0.86 EGFR (0.68) STK4SRCEGFRERBB2
SCHEMBL15320486 0.86 MAP2K1 (0.72) STK4EGFRERBB2MAP2K1
SCHEMBL22419601 0.84 EGFR (0.71) STK4SRCEGFRERBB2
SCHEMBL28547991 0.84 EGFR (0.64) STK4EGFRERBB2MAP2K1
SCHEMBL27974765 0.83 EGFR (0.62) STK4SRCEGFRERBB2MAP2K1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112759583-B Quinoline derivative containing furyl and preparation method and application thereof 河南省医药科学研究院 2022-10-11 CN disclosed
CN-112694439-B Phenyl acrylamide quinoline derivative and preparation method and application thereof 河南省医药科学研究院 2022-08-30 CN disclosed
CN-112625025-B Pyridyl substituted quinoline derivative and its prepn and use 河南省医药科学研究院 2022-03-29 CN disclosed
CN-112759583-A Quinoline derivative containing furyl and preparation method and application thereof 河南省医药科学研究院 2021-05-07 CN disclosed
CN-112694439-A Phenyl acrylamide quinoline derivative and preparation method and application thereof 河南省医药科学研究院 2021-04-23 CN disclosed
CN-112625025-A Pyridyl substituted quinoline derivative and its prepn and use 河南省医药科学研究院 2021-04-09 CN disclosed