SCHEMBL2855574

SCHEMBL2855574

NC(=O)C1C[CH]CCN1Cc1cccc(Cl)c1

nearest known ligand 0.46

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
SPHK1 Q9NYA1 1/20 0.44
SIGMAR1 Q99720 1/20 0.43
KMT2A Q03164 1/20 0.43
MAOA P21397 3/20 0.43
MAOB P27338 3/20 0.43
TDP1 Q9NUW8 1/20 0.43
DRD4 P21917 1/20 0.43
MAPT P10636 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
ADRA1D P25100 1/20 0.42
NPBWR1 P48145 1/20 0.42
MCHR1 Q99705 1/20 0.42
ATM Q13315 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
AMPD2 Q01433 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2699801 0.87 SPHK1 (0.49) SPHK1MAOAMAOBCYP2C19
SCHEMBL14142405 0.85 GAA (0.46) KDM4ESPHK1MAOAMAOBDRD4
SCHEMBL7309417 0.82 SPHK1 (0.63) KDM4ESPHK1MAOAMAOBTDP1
SCHEMBL6501382 0.81 KMT2A (0.54) KDM4ESPHK1KMT2AMAOAMAOB
SCHEMBL6505049 0.81 FAAH (0.48) SPHK1KMT2AMAOAMAOB
SCHEMBL4704664 0.79 GBA1 (0.40) KDM4ESPHK1SIGMAR1KMT2AMAOA
SCHEMBL2852932 0.79 MAOB (0.47) SPHK1MAOAMAOB
SCHEMBL4592233 0.79 SPHK1 (0.40) KDM4ESPHK1SIGMAR1KMT2AMAOA
SCHEMBL5015327 0.78 KDM4E (0.48) KDM4ESIGMAR1DRD4MAPT
SCHEMBL6504152 0.77 CCR8 (0.52) SPHK1KMT2AMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed