SCHEMBL2855705

SCHEMBL2855705

COc1ccc(-n2ncc(C(=O)NCc3ccc(Cl)c(Cl)c3)c2C(F)(F)F)cc1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 6/20 0.56
TRPC3 Q13507 1/20 0.51
DGAT2 Q96PD7 1/20 0.49
APEX1 P27695 1/20 0.49
TP53 P04637 3/20 0.49
RPA1 P27694 2/20 0.47
SMO Q99835 1/20 0.47
KDM4E B2RXH2 1/20 0.46
ALDH1A1 P00352 1/20 0.46
THRB P10828 1/20 0.46
DDR1 Q08345 1/20 0.46
MAPK11 Q15759 1/20 0.46
MAPK14 Q16539 1/20 0.46
DDR2 Q16832 1/20 0.46
TMEM97 Q5BJF2 1/20 0.46
MAP3K20 Q9NYL2 1/20 0.46
MAP3K2 Q9Y2U5 1/20 0.46
NR3C1 P04150 1/20 0.45
POLB P06746 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2859678 0.89 CCR1 (0.55) CCR1TRPC3DGAT2TP53ALDH1A1
SCHEMBL2854425 0.89 CCR1 (0.60) CCR1TRPC3KDM4EALDH1A1DDR1
SCHEMBL2858070 0.88 CCR1 (0.57) CCR1TRPC3TP53SMOKDM4E
SCHEMBL2860317 0.88 CCR1 (0.62) CCR1TRPC3KDM4EALDH1A1DDR1
SCHEMBL2857636 0.87 KDM4E (0.61) CCR1TRPC3DGAT2KDM4EALDH1A1
SCHEMBL2855224 0.86 CCR1 (0.55) CCR1DGAT2TP53KDM4EALDH1A1
SCHEMBL2855701 0.85 CCR1 (0.54) CCR1TRPC3DGAT2TP53KDM4E
SCHEMBL2850316 0.85 TP53 (0.59) CCR1DGAT2TP53KDM4EALDH1A1
SCHEMBL2856625 0.85 TSHR (0.48) CCR1RPA1SMO
SCHEMBL2854971 0.85 CCR1 (0.66) CCR1DGAT2KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed