SCHEMBL2858070

SCHEMBL2858070

O=C(NCc1ccc(Cl)c(Cl)c1)c1cnn(-c2ccc(F)cc2)c1C(F)(F)F

nearest known ligand 0.57

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 10/20 0.57
MAPK1 P28482 1/20 0.55
P2RX7 Q99572 1/20 0.54
TRPC3 Q13507 1/20 0.52
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
SMO Q99835 2/20 0.48
DDR1 Q08345 1/20 0.48
MAPK11 Q15759 1/20 0.48
MAPK14 Q16539 1/20 0.48
DDR2 Q16832 1/20 0.48
TMEM97 Q5BJF2 1/20 0.48
MAP3K20 Q9NYL2 1/20 0.48
MAP3K2 Q9Y2U5 1/20 0.48
TP53 P04637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854425 0.93 CCR1 (0.60) CCR1MAPK1TRPC3KDM4EALDH1A1
SCHEMBL2860317 0.92 CCR1 (0.62) CCR1MAPK1P2RX7TRPC3KDM4E
SCHEMBL2857636 0.91 KDM4E (0.61) CCR1P2RX7TRPC3KDM4EALDH1A1
SCHEMBL2856181 0.89 CCR1 (0.56) CCR1P2RX7TRPC3KDM4EALDH1A1
SCHEMBL2855705 0.88 CCR1 (0.56) CCR1TRPC3KDM4EALDH1A1SMO
SCHEMBL2860444 0.88 CCR1 (0.60) CCR1MAPK1TRPC3KDM4EALDH1A1
SCHEMBL2850548 0.85 CCR1 (0.61) CCR1TRPC3KDM4EALDH1A1SMO
SCHEMBL2857923 0.84 CCR1 (0.66) CCR1P2RX7TRPC3KDM4EALDH1A1
SCHEMBL2857342 0.84 CCR1 (0.60) CCR1TRPC3KDM4EALDH1A1DDR1
SCHEMBL2852102 0.84 ALDH1A1 (0.67) CCR1KDM4EALDH1A1SMODDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed