SCHEMBL2850316

SCHEMBL2850316

COc1ccc(-n2ncc(C(=O)NCc3ccccc3)c2C(F)(F)F)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 4/20 0.59
ALDH1A1 P00352 4/20 0.58
KDM4E B2RXH2 3/20 0.58
HPGD P15428 2/20 0.57
DGAT2 Q96PD7 2/20 0.57
DDR1 Q08345 1/20 0.55
MAPK11 Q15759 1/20 0.55
MAPK14 Q16539 1/20 0.55
DDR2 Q16832 1/20 0.55
TMEM97 Q5BJF2 1/20 0.55
MAP3K20 Q9NYL2 1/20 0.55
MAP3K2 Q9Y2U5 1/20 0.55
CNR2 P34972 1/20 0.55
MAPT P10636 4/20 0.53
SMN1; SMN2 Q16637 2/20 0.52
POLB P06746 1/20 0.52
CCR1 P32246 2/20 0.51
NR3C1 P04150 1/20 0.51
NPSR1 Q6W5P4 1/20 0.50
LMNA P02545 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855224 0.91 CCR1 (0.55) TP53ALDH1A1KDM4EDGAT2DDR1
SCHEMBL2859678 0.90 CCR1 (0.55) TP53ALDH1A1DGAT2DDR1MAPK11
SCHEMBL2855239 0.90 ALDH1A1 (0.56) TP53ALDH1A1KDM4EHPGDDGAT2
SCHEMBL2854971 0.89 CCR1 (0.66) KDM4EDGAT2POLBCCR1NPSR1
SCHEMBL2860213 0.89 KDM4E (0.73) ALDH1A1KDM4EHPGDDGAT2DDR1
SCHEMBL2855701 0.88 CCR1 (0.54) TP53ALDH1A1KDM4EDGAT2DDR1
SCHEMBL2850153 0.87 KDM4E (0.63) ALDH1A1KDM4EHPGDDDR1MAPK11
SCHEMBL2852896 0.87 KDM4E (0.63) TP53ALDH1A1KDM4EHPGDDDR1
SCHEMBL2852015 0.86 CCR1 (0.63) ALDH1A1KDM4EHPGDDDR1MAPK11
SCHEMBL10366447 0.86 TRPC3 (0.62) TP53ALDH1A1KDM4EHPGDDGAT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed