SCHEMBL28560847

SCHEMBL28560847

CCCNc1c(N)cc(C(N)=O)cc1OCCC1CN(C(=O)OC(C)(C)C)C1

nearest known ligand 0.38

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 2/20 0.38
SCN9A Q15858 1/20 0.38
JAK3 P52333 1/20 0.36
NAMPT P43490 1/20 0.35
PDE4B Q07343 3/20 0.35
NR1H2 P55055 1/20 0.35
GPR119 Q8TDV5 4/20 0.34
USP30 Q70CQ3 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC2 Q92769 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
HTR6 P50406 3/20 0.33
BCHE P06276 2/20 0.33
ALOX5AP P20292 1/20 0.33
FEN1 P39748 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28557043 0.91 CHEK2 (0.38) CHEK2SCN9ANAMPTPDE4BNR1H2
SCHEMBL28556407 0.87 MAPT (0.36) CHEK2SCN9AJAK3NAMPTPDE4B
SCHEMBL22857826 0.86 SCN9A (0.42) CHEK2SCN9APDE4BGPR119USP30
SCHEMBL28560849 0.82 PDE4D (0.35) NAMPTPDE4BNR1H2GPR119USP30
SCHEMBL21158729 0.81 TSHR (0.35)
SCHEMBL22857887 0.79 STING1 (0.42) SCN9A
SCHEMBL28548767 0.78 MAPT (0.37) CHEK2SCN9ANAMPTPDE4BNR1H2
SCHEMBL22857866 0.78 STING1 (0.46)
SCHEMBL22121045 0.78 TSHR (0.43)
SCHEMBL22857823 0.77 CA12 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110016021-B Immunomodulator 成都先导药物开发股份有限公司 2021-05-07 CN disclosed