SCHEMBL21158729

SCHEMBL21158729

CCCNc1c(N)cc(C(N)=O)cc1OCCC1COC1

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.35
ALDH1A1 P00352 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
STING1 Q86WV6 2/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31
BPTF Q12830 1/20 0.31
CREBBP Q92793 1/20 0.31
MAPK1 P28482 1/20 0.30
PTGER4 P35408 1/20 0.30
PPARG P37231 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21158913 0.91 USP2 (0.33) TSHRALDH1A1SMN1; SMN2CREBBPPTGER4
SCHEMBL21158909 0.89 IRAK4 (0.38) TSHRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL28548646 0.85 MAPT (0.41) ALDH1A1SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL22121045 0.84 TSHR (0.43) TSHRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL21158643 0.82 STING1 (0.42) TSHRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL21158654 0.81 PARP15 (0.43) TSHRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL28560847 0.81 CHEK2 (0.38)
SCHEMBL21158981 0.80 TSHR (0.34) TSHRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL21158926 0.77 SMN1; SMN2 (0.36) TSHRALDH1A1SMN1; SMN2MEN1KMT2A
SCHEMBL21158773 0.77 PDE4D (0.50)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110016021-B Immunomodulator 成都先导药物开发股份有限公司 2021-05-07 CN disclosed
WO-2019134707-A1 IMMUNOMODULATOR 成都先导药物开发股份有限公司 2019-07-11 WO disclosed