SCHEMBL28566737

SCHEMBL28566737

NC(=O)Oc1ccc(OCc2ccnc(Nc3cnc(C(=O)NCCO)cn3)c2)c2ccccc12

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GPR52 Q9Y2T5 15/20 0.40
MAPK14 Q16539 2/20 0.36
HTR2B P41595 1/20 0.35
BRD4 O60885 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
HCK P08631 1/20 0.34
MAPK12 P53778 1/20 0.34
SPHK2 Q9NRA0 1/20 0.34
SPHK1 Q9NYA1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17008512 0.91 GPR52 (0.41) GPR52MAPK14HTR2BBRD4MRGPRX4
SCHEMBL18567061 0.89 GPR52 (0.44) GPR52MAPK14HTR2BBRD4HCK
SCHEMBL17008514 0.86 MAPK14 (0.46) GPR52MAPK14BRD4HCKMAPK12
SCHEMBL17008486 0.83 MAPK14 (0.44) GPR52MAPK14MRGPRX4HCKMAPK12
SCHEMBL28588449 0.82 LRRK2 (0.45) MAPK14MRGPRX4HCKMAPK12
SCHEMBL17017553 0.82 MAPK14 (0.44) GPR52MAPK14BRD4HCKMAPK12
SCHEMBL28578481 0.79 HCK (0.39) MAPK14MRGPRX4HCKMAPK12
SCHEMBL17017129 0.79 MRGPRX4 (0.40) MAPK14MRGPRX4HCKMAPK12
SCHEMBL17008525 0.78 MAPK14 (0.42) GPR52MAPK14MRGPRX4HCKMAPK12
SCHEMBL31086537 0.78 MAPK14 (0.42) GPR52MAPK14MRGPRX4HCKMAPK12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113264921-A Pyrazolyl-ureas as kinase inhibitors 瑞斯比维特有限公司 2021-08-17 CN disclosed
CN-106573914-B Pyrazolyl-ureas as kinase inhibitors 瑞斯比维特有限公司 2021-05-28 CN disclosed