SCHEMBL28566754

SCHEMBL28566754

Cc1cc(C(=O)OC(C)C)cc2sc(Br)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 4/20 0.44
CA1 P00915 4/20 0.44
CA2 P00918 4/20 0.44
CA7 P43166 4/20 0.44
CA9 Q16790 4/20 0.44
CA14 Q9ULX7 4/20 0.44
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
LCK P06239 1/20 0.38
ALDH1A1 P00352 4/20 0.38
L3MBTL1 Q9Y468 1/20 0.36
MAPK1 P28482 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
PTPN11 Q06124 2/20 0.36
GAA P10253 1/20 0.35
USP2 O75604 1/20 0.35
PDCD1 Q15116 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28570422 0.85 HSD17B10 (0.51) CA12CA1CA2CA7CA9
SCHEMBL9957845 0.84 PIK3CA (0.44) CA12CA1CA2CA7CA9
SCHEMBL21925010 0.79 NPC1 (0.41) NPC1RAB9ALCKALDH1A1KDM4E
SCHEMBL21062982 0.73 NPC1 (0.43) CA12CA1CA2CA7CA9
SCHEMBL23730805 0.72 NPC1 (0.44) CA12CA1CA2CA7CA9
SCHEMBL29644660 0.71 ALDH1A1 (0.45) CA12CA1CA2CA7CA9
SCHEMBL9955853 0.71 ALDH1A1 (0.45) CA12CA1CA2CA7CA9
SCHEMBL22922699 0.70 LCK (0.46) MEN1KMT2ANPC1RAB9ALCK
SCHEMBL20094458 0.70 ALDH1A1 (0.45) CA12CA1CA2CA7CA9
SCHEMBL3644443 0.70 CA12 (0.45) CA12CA1CA2CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109265471-B FXR receptor agonists 轩竹生物科技有限公司 2021-06-04 CN disclosed