SCHEMBL28567710

SCHEMBL28567710

Cc1ccccc1-c1nc(C(=O)O)cc2c1[nH]c1ccccc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 9/20 0.58
MEN1 O00255 8/20 0.58
MGAM O43451 7/20 0.53
KDM4E B2RXH2 2/20 0.52
MAPT P10636 2/20 0.52
LMNA P02545 2/20 0.52
ALDH1A1 P00352 1/20 0.52
TP53 P04637 1/20 0.52
HPGD P15428 1/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52
GABRP O00591 1/20 0.49
GABRD O14764 1/20 0.49
GABRA1 P14867 1/20 0.49
GABRB1 P18505 1/20 0.49
GABRG2 P18507 1/20 0.49
GABRB3 P28472 1/20 0.49
GABRA5 P31644 1/20 0.49
GABRA3 P34903 1/20 0.49
GABRA2 P47869 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28558217 0.86 KMT2A (0.55) KMT2AMEN1MGAMKDM4EMAPT
SCHEMBL27963004 0.85 HDAC3 (0.61) KMT2AMEN1MGAMKDM4EMAPT
SCHEMBL30607054 0.85 HDAC3 (0.61) KMT2AMEN1MGAMKDM4EMAPT
SCHEMBL28556004 0.84 KMT2A (0.53) KMT2AMEN1MGAMKDM4EMAPT
SCHEMBL27917533 0.84 MEN1 (0.74) KMT2AMEN1MGAM
Harman-3-Carboxylic Acid SCHEMBL3967948 0.82 MAPT (0.73) KMT2AMEN1KDM4EMAPTLMNA
SCHEMBL30607047 0.82 HDAC1 (0.53) KMT2AMEN1MGAMKDM4EMAPT
SCHEMBL2216422 0.80 MEN1 (0.65) KMT2AMEN1MGAMPOLBMITF
SCHEMBL30607046 0.79 MGAM (0.57) KMT2AMEN1MGAMKDM4EMAPT
SCHEMBL29817694 0.79 MEN1 (0.63) KMT2AMEN1MGAMPOLBMITF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109134460-B Synthesis method of beta-carboline compound 南开大学 2021-04-06 CN disclosed