SCHEMBL28568849

SCHEMBL28568849

O=S1(=O)CCC(c2ccc(Br)cc2)N1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 6/20 0.40
MAOB P27338 3/20 0.40
ALDH1A1 P00352 1/20 0.36
CYP3A4 P08684 3/20 0.35
CYP2C9 P11712 3/20 0.35
CYP2C19 P33261 2/20 0.35
LMNA P02545 1/20 0.35
TSHR P16473 1/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35
KCNH2 Q12809 2/20 0.34
RCOR1 Q9UKL0 2/20 0.34
KDM1B Q8NB78 1/20 0.34
SMN1; SMN2 Q16637 2/20 0.33
MAPT P10636 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
GALR1 P47211 1/20 0.33
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
MEN1 O00255 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28297380 0.81 KCNH2 (0.37) KDM1AALDH1A1TSHRKCNH2SMN1; SMN2
SCHEMBL14686714 0.81 MEN1 (0.37) SMN1; SMN2MEN1KMT2A
SCHEMBL738878 0.81 MEN1 (0.37) SMN1; SMN2MEN1KMT2A
SCHEMBL28325770 0.78 ALDH1A1 (0.36) KDM1AMAOBALDH1A1CYP3A4CYP2C9
SCHEMBL28325760 0.77 DDB1 (0.42) KDM1AMAOBALDH1A1SMN1; SMN2MAPT
SCHEMBL4065116 0.71 KDM1A (0.38) KDM1AMAOBKCNH2RCOR1KDM1B
SCHEMBL5187861 0.70 MEN1 (0.36) SMN1; SMN2MEN1KMT2A
SCHEMBL5877853 0.70 KDM1A (0.37) KDM1AMAOBCYP3A4CYP2C9CYP2C19
SCHEMBL2756273 0.70 KDM1A (0.40) KDM1AMAOBALDH1A1CYP3A4CYP2C9
SCHEMBL20401774 0.69 KDM1A (0.43) KDM1AMAOBALDH1A1CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110372628-B Internal sulfonamide compound and preparation method thereof 武汉大学 2021-04-02 CN disclosed