SCHEMBL28569264

SCHEMBL28569264

COC(=O)C(Cc1c(C)cc(O)cc1C)NC(=O)OC(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KLK5 Q9Y337 1/20 0.47
CTSS P25774 4/20 0.43
CTSK P43235 2/20 0.43
TACR1 P25103 2/20 0.42
ACE P12821 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
MAPT P10636 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MDM4 O15151 1/20 0.39
MDM2 Q00987 1/20 0.39
PPARA Q07869 1/20 0.39
MAP1LC3B Q9GZQ8 1/20 0.39
MAP1LC3A Q9H492 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23375845 1.00 KLK5 (0.47) KLK5CTSSCTSKTACR1ACE
SCHEMBL10759759 0.88 KLK5 (0.47) KLK5CTSSCTSKTACR1ACE
SCHEMBL21029360 0.88 KLK5 (0.47) KLK5CTSSCTSKTACR1ACE
SCHEMBL1055585 0.88 ACE (0.52) CTSSCTSKACECTSLCTSB
SCHEMBL2263756 0.88 ACE (0.52) CTSSCTSKACECTSLCTSB
SCHEMBL12294697 0.88 CTSS (0.44) CTSSCTSKTACR1ACECTSL
SCHEMBL13252065 0.87 KLK5 (0.46) KLK5CTSSCTSKTACR1ACE
SCHEMBL1061605 0.87 KLK5 (0.48) KLK5CTSSCTSKTACR1ACE
SCHEMBL1061604 0.87 KLK5 (0.48) KLK5CTSSCTSKTACR1ACE
SCHEMBL1056766 0.86 KLK5 (0.45) KLK5CTSSCTSKTACR1ACE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112867705-A Opioid receptor modulators and products and methods related thereto 埃皮欧黛公司 2021-05-28 CN disclosed