SCHEMBL28573045

SCHEMBL28573045

O=C(O)c1cccnc1CNCc1ccncc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 6/20 0.46
KDM4E B2RXH2 3/20 0.45
TDP1 Q9NUW8 1/20 0.45
ALDH1A1 P00352 3/20 0.44
SLC2A4 P14672 1/20 0.44
MAPT P10636 2/20 0.44
CYP3A4 P08684 1/20 0.44
ALOX15 P16050 1/20 0.44
TSHR P16473 1/20 0.44
BLM P54132 1/20 0.44
AGER Q15109 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
MAPK1 P28482 1/20 0.43
KDM6B O15054 1/20 0.43
KDM4A O75164 1/20 0.43
KDM4D Q6B0I6 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
GAA P10253 1/20 0.43
NAPRT Q6XQN6 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28109150 0.82 ALDH1A1 (0.54) KDM4EALDH1A1MAPTNPSR1LMNA
SCHEMBL2129251 0.79 SMN1; SMN2 (0.49) KDRKDM4ETDP1ALDH1A1MAPT
SCHEMBL27648140 0.79 ALDH1A1 (0.49) KDM4EALDH1A1SLC2A4MAPTMAPK1
SCHEMBL1715372 0.78 KDR (0.65) KDRKDM4EKDM6BKDM4AKDM4D
SCHEMBL4431043 0.74 KDM4E (0.49) KDM4ETDP1ALDH1A1MAPTCYP3A4
SCHEMBL3880000 0.72 KDM4E (0.59) KDM4ETDP1ALDH1A1MAPTCYP3A4
SCHEMBL5252687 0.72 KDM4E (0.59) KDM4ETDP1ALDH1A1MAPTCYP3A4
SCHEMBL258223 0.71 ALDH1A1 (0.55) KDM4ETDP1ALDH1A1MAPTCYP3A4
SCHEMBL1042566 0.71 SLC2A4 (0.63) TDP1ALDH1A1SLC2A4MAPTGAA
SCHEMBL1722473 0.71 SMN1; SMN2 (0.57) KDM4ETDP1ALDH1A1MAPTCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108467360-B Preparation method and intermediate of apatinib 江苏美迪克化学品有限公司 2021-04-30 CN disclosed