SCHEMBL28575652

SCHEMBL28575652

C[SiH](C)OC(c1ccccn1)C(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 2/20 0.39
SLC6A2 P23975 2/20 0.39
SLC6A4 P31645 2/20 0.39
TSHR P16473 2/20 0.39
KCNA5 P22460 5/20 0.37
KCNH2 Q12809 1/20 0.37
CYP2C19 P33261 1/20 0.35
KCNE1 P15382 2/20 0.35
CYP2D6 P10635 1/20 0.35
CYP3A4 P08684 2/20 0.35
KDM4E B2RXH2 2/20 0.35
LMNA P02545 2/20 0.35
ABCB11 O95342 1/20 0.35
ESR1 P03372 1/20 0.35
ADRA2A P08913 1/20 0.35
CYP2C9 P11712 1/20 0.35
PDE4A P27815 1/20 0.35
ADRA1A P35348 1/20 0.35
OPRK1 P41145 1/20 0.35
STAT6 P42226 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7448598 0.82 SLC6A3 (0.44) SLC6A3SLC6A2SLC6A4TSHRKCNA5
SCHEMBL21742268 0.80 TSHR (0.46) SLC6A3SLC6A2SLC6A4TSHRKCNA5
SCHEMBL21742017 0.76 KCNH2 (0.44) SLC6A3SLC6A2SLC6A4TSHRKCNA5
SCHEMBL15277627 0.75 TSHR (0.41) SLC6A3SLC6A2SLC6A4TSHRKCNA5
SCHEMBL28528911 0.75
SCHEMBL21742152 0.73 TSHR (0.49) SLC6A3SLC6A2SLC6A4TSHRCYP2C19
SCHEMBL507789 0.73 GBA1 (0.31)
SCHEMBL5719027 0.73 IRAK4 (0.38)
SCHEMBL3387686 0.73 KDM4E (0.36) KDM4E
SCHEMBL5465600 0.72 NOS3 (0.38) TSHRKDM4ELMNAHIF1AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107709301-B Pyrazole derivative or pharmacologically acceptable salt thereof 橘生药品工业株式会社 2021-06-22 CN disclosed