SCHEMBL2857713

SCHEMBL2857713

CS(=O)(=O)c1cccc(C(=O)Nc2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)c1

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.49
ALDH1A1 P00352 3/20 0.47
RXFP1 Q9HBX9 1/20 0.47
SIRT2 Q8IXJ6 3/20 0.44
NPC1 O15118 2/20 0.44
RAB9A P51151 2/20 0.44
TSHR P16473 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
MAPT P10636 1/20 0.43
LMNA P02545 2/20 0.42
TDP1 Q9NUW8 1/20 0.42
ORAI1 Q96D31 1/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
EGFR P00533 1/20 0.41
FGFR1 P11362 1/20 0.41
KDR P35968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2854048 0.86 MAPT (0.50) CCR1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL2852110 0.85 SMN1; SMN2 (0.54) ALDH1A1NPC1RAB9ATSHRSMN1; SMN2
SCHEMBL8631115 0.84 KMT2A (0.49) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL2856664 0.83 CYP1A2 (0.55) ALDH1A1RXFP1NPC1RAB9ASMN1; SMN2
SCHEMBL2859981 0.83 KDM4E (0.50) ALDH1A1NPC1RAB9ASMN1; SMN2MAPT
SCHEMBL13513684 0.81 CCR1 (0.54) CCR1ALDH1A1MAPTMEN1KMT2A
SCHEMBL14539381 0.79 CCR1 (0.42) CCR1ALDH1A1NPC1RAB9AMAPT
SCHEMBL2855798 0.77 MAPT (0.45) CCR1ALDH1A1SMN1; SMN2MAPTLMNA
SCHEMBL2858063 0.76 MAPT (0.57) CCR1ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL8630975 0.76 PTGS2 (0.59) ALDH1A1SMN1; SMN2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed