SCHEMBL2856664

SCHEMBL2856664

COc1cccc(C(=O)Nc2cnn(-c3ccc(Cl)cc3)c2C(F)(F)F)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C19 P33261 1/20 0.55
RAB9A P51151 5/20 0.51
NPC1 O15118 3/20 0.51
GAA P10253 2/20 0.51
ALDH1A1 P00352 2/20 0.51
SMN1; SMN2 Q16637 5/20 0.50
MAPT P10636 4/20 0.50
LMNA P02545 3/20 0.50
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
THRB P10828 1/20 0.49
POLB P06746 3/20 0.49
ADORA2A P29274 1/20 0.49
ADORA1 P30542 1/20 0.49
HTT P42858 1/20 0.49
KDM4E B2RXH2 1/20 0.48
KCNQ3 O43525 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852110 0.86 SMN1; SMN2 (0.54) RAB9ANPC1ALDH1A1SMN1; SMN2MAPT
SCHEMBL2859981 0.84 KDM4E (0.50) CYP1A2CYP2D6CYP2C19RAB9ANPC1
SCHEMBL2857713 0.83 CCR1 (0.49) RAB9ANPC1ALDH1A1SMN1; SMN2MAPT
SCHEMBL2860020 0.80 KDM4E (0.51) RAB9ANPC1GAAALDH1A1SMN1; SMN2
SCHEMBL2859050 0.80 PTGS1 (0.46) CYP1A2CYP3A4CYP2C19RAB9ANPC1
SCHEMBL2859651 0.77 MAPT (0.46) RAB9ANPC1ALDH1A1SMN1; SMN2MAPT
SCHEMBL2858063 0.77 MAPT (0.57) RAB9ANPC1ALDH1A1SMN1; SMN2MAPT
SCHEMBL2858311 0.77 RAB9A (0.47) CYP3A4CYP2C19RAB9ANPC1ALDH1A1
SCHEMBL2854156 0.76 ROCK2 (0.46) CYP1A2CYP3A4CYP2D6CYP2C19RAB9A
SCHEMBL2856049 0.76 ATM (0.53) RAB9ANPC1ALDH1A1SMN1; SMN2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed