SCHEMBL28577166

SCHEMBL28577166

CCOC(=O)C(C)(C)C1CCN(C(=O)N2CCN(C(=O)OC(C)(C)C)CC2)CC1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
RECQL P46063 2/20 0.44
HPGD P15428 1/20 0.44
EPHX1 P07099 1/20 0.42
GPR119 Q8TDV5 3/20 0.41
KDM4E B2RXH2 1/20 0.41
MAPT P10636 1/20 0.41
THRB P10828 1/20 0.41
GAA P10253 1/20 0.41
HRH3 Q9Y5N1 2/20 0.41
ALDH1A1 P00352 3/20 0.40
MEN1 O00255 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40
USP2 O75604 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
CYP2D6 P10635 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19995830 0.95 HPGD (0.48) RECQLHPGDEPHX1GPR119KDM4E
SCHEMBL22680079 0.86 GAA (0.43) RECQLHPGDEPHX1GPR119MAPT
SCHEMBL22680073 0.86 GAA (0.43) RECQLHPGDEPHX1GPR119MAPT
SCHEMBL22680078 0.86 GAA (0.43) RECQLHPGDEPHX1GPR119MAPT
SCHEMBL28577921 0.82 HPGD (0.49) RECQLHPGDEPHX1GPR119KDM4E
SCHEMBL30659463 0.81 HPGD (0.46) RECQLHPGDEPHX1GPR119KDM4E
SCHEMBL8329687 0.80 GPR119 (0.45) RECQLHPGDEPHX1GPR119GAA
SCHEMBL18285469 0.79 EPHX1 (0.52) RECQLHPGDEPHX1GPR119KDM4E
SCHEMBL2319139 0.79 GAA (0.41) MAPTTHRBGAAALDH1A1MEN1
SCHEMBL1189317 0.78 ALDH1A1 (0.56) RECQLHPGDKDM4EMAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112778299-B Piperazine ureido derivatives, preparation method thereof and application thereof in medicines 江苏恒瑞医药股份有限公司 2023-07-14 CN disclosed
CN-112778299-A Piperazine ureido derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-05-11 CN disclosed