SCHEMBL2857735

SCHEMBL2857735

O=C(NCCc1cccc(C(F)(F)F)c1)Oc1cnn(-c2ccc(Cl)cc2)c1C(F)(F)F

nearest known ligand 0.54

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 13/20 0.54
CNR1 P21554 1/20 0.52
NPSR1 Q6W5P4 2/20 0.51
HSP90AA1 P07900 1/20 0.51
MAPT P10636 1/20 0.51
TRPV1 Q8NER1 1/20 0.42
TAAR1 Q96RJ0 1/20 0.42
KDM4E B2RXH2 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2852505 0.93 ABCB1 (0.48) CCR1CNR1NPSR1HSP90AA1MAPT
SCHEMBL2854340 0.92 CCR1 (0.53) CCR1CNR1NPSR1HSP90AA1MAPT
SCHEMBL2863198 0.92 CCR1 (0.50) CCR1CNR1NPSR1MAPTTRPV1
SCHEMBL2857238 0.91 CCR1 (0.43) CCR1CNR1NPSR1HSP90AA1MAPT
SCHEMBL2858011 0.91 ABCB1 (0.51) CCR1CNR1NPSR1HSP90AA1MAPT
SCHEMBL2849956 0.91 CCR1 (0.62) CCR1NPSR1HSP90AA1MAPT
SCHEMBL2855547 0.90 TAAR1 (0.54) CCR1CNR1NPSR1HSP90AA1MAPT
SCHEMBL2863131 0.89 CNR1 (0.50) CCR1CNR1NPSR1HSP90AA1MAPT
SCHEMBL2860669 0.89 TAAR1 (0.46) CCR1CNR1MAPTTAAR1KDM4E
SCHEMBL2860847 0.88 CCR1 (0.55) CCR1CNR1NPSR1HSP90AA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed