SCHEMBL28577368

SCHEMBL28577368

COC(=O)[C@H]1CCCN(C(=O)N2CCN(C(=O)OC(C)(C)C)CC2)C1

nearest known ligand 0.53

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.53
ALDH1A1 P00352 2/20 0.52
MEN1 O00255 1/20 0.52
MAPT P10636 1/20 0.52
KMT2A Q03164 1/20 0.52
EPHX1 P07099 1/20 0.48
HRH3 Q9Y5N1 1/20 0.44
ABL1 P00519 1/20 0.44
RIN1 Q13671 1/20 0.44
SMN1; SMN2 Q16637 2/20 0.43
RECQL P46063 1/20 0.42
PTPN2 P17706 1/20 0.41
PTPN1 P18031 1/20 0.41
PTPN6 P29350 1/20 0.41
STS P08842 1/20 0.41
EPHX2 P34913 1/20 0.40
USP2 O75604 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28574242 1.00 HPGD (0.53) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL28574240 1.00 HPGD (0.53) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL641371 0.90 ALDH1A1 (0.61) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL641372 0.90 ALDH1A1 (0.61) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL9882415 0.90 ALDH1A1 (0.61) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL28914926 0.86 HPGD (0.56) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL28571024 0.86 HPGD (0.56) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL22570055 0.86 HPGD (0.59) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL28571023 0.86 HPGD (0.56) HPGDALDH1A1MEN1MAPTKMT2A
SCHEMBL23210360 0.86 HPGD (0.58) HPGDALDH1A1MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112778299-B Piperazine ureido derivatives, preparation method thereof and application thereof in medicines 江苏恒瑞医药股份有限公司 2023-07-14 CN disclosed
CN-112778299-A Piperazine ureido derivative, preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-05-11 CN disclosed