SCHEMBL28577446

SCHEMBL28577446

COc1ccccc1Oc1c(Cl)nc(-c2cccc(Cl)c2)nc1Cl

nearest known ligand 0.83

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DHPS P49366 17/20 0.83
TSHR P16473 2/20 0.52
NPC1 O15118 1/20 0.52
MAPT P10636 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
NR1I3 Q14994 1/20 0.51
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28577292 0.91 DHPS (1.00) DHPS
SCHEMBL30412354 0.91 DHPS (1.00) DHPS
SCHEMBL28587165 0.88 DHPS (0.84) DHPSTSHRNPC1SMN1; SMN2MEN1
SCHEMBL7851372 0.88 DHPS (0.84) DHPSMAPTSMN1; SMN2NR1I3
SCHEMBL7303389 0.87 DHPS (0.81) DHPSMAPTMEN1KMT2A
SCHEMBL30450864 0.86 DHPS (0.84) DHPS
SCHEMBL28589425 0.86 DHPS (0.84) DHPS
SCHEMBL28584109 0.86 DHPS (0.65) DHPS
SCHEMBL28589605 0.84 DHPS (0.82) DHPS
SCHEMBL6964288 0.83 DHPS (0.61) DHPSTSHRMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112898208-B Phenylpyrimidine amine antitumor compound and preparation method and application thereof 中国医科大学 2023-06-20 CN disclosed
CN-112898208-A Phenyl pyrimidinamine antitumor compound and preparation method and application thereof 中国医科大学 2021-06-04 CN disclosed