SCHEMBL28587165

SCHEMBL28587165

COc1ccccc1Oc1c(Cl)nc(-c2cccc(C)c2)nc1Cl

nearest known ligand 0.84

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHPS P49366 15/20 0.84
SMN1; SMN2 Q16637 3/20 0.51
HSD17B10 Q99714 3/20 0.51
ALDH1A1 P00352 3/20 0.51
HPGD P15428 3/20 0.51
TP53 P04637 2/20 0.51
NPC1 O15118 2/20 0.51
RAB9A P51151 2/20 0.51
MEN1 O00255 2/20 0.51
KMT2A Q03164 2/20 0.51
NFKB1 P19838 1/20 0.51
NFKB2 Q00653 1/20 0.51
RELA Q04206 1/20 0.51
KDM4E B2RXH2 2/20 0.49
TSHR P16473 2/20 0.49
POLB P06746 1/20 0.48
LMNA P02545 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30411986 0.91 DHPS (1.00) DHPS
SCHEMBL28566926 0.91 DHPS (1.00) DHPS
SCHEMBL28577446 0.88 DHPS (0.83) DHPSSMN1; SMN2NPC1MEN1KMT2A
SCHEMBL7851372 0.86 DHPS (0.84) DHPSSMN1; SMN2
SCHEMBL7303389 0.86 DHPS (0.81) DHPSALDH1A1MEN1KMT2ALMNA
SCHEMBL28589425 0.85 DHPS (0.84) DHPS
SCHEMBL28584109 0.85 DHPS (0.65) DHPS
SCHEMBL30450864 0.85 DHPS (0.84) DHPS
SCHEMBL28584053 0.85 DHPS (0.82) DHPSTSHRLMNA
SCHEMBL6964288 0.82 DHPS (0.61) DHPSALDH1A1MEN1KMT2ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112898208-B Phenylpyrimidine amine antitumor compound and preparation method and application thereof 中国医科大学 2023-06-20 CN disclosed
CN-112898208-A Phenyl pyrimidinamine antitumor compound and preparation method and application thereof 中国医科大学 2021-06-04 CN disclosed