SCHEMBL28579656

SCHEMBL28579656

C=CC(=O)Nc1ccc(OC)c(Nc2ncc(Cl)c(Nc3ccc(N4CCN(C(C)=O)CC4)cc3OC)n2)c1

nearest known ligand 0.83

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
EGFR P00533 5/20 0.83
MAPK3 P27361 2/20 0.81
ALK Q9UM73 13/20 0.77

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28595246 0.94 MAPK3 (0.81) EGFRMAPK3ALK
SCHEMBL28053891 0.92 JAK3 (0.77) EGFRMAPK3ALK
SCHEMBL2724456 0.91 EGFR (1.00) EGFRMAPK3ALK
SCHEMBL28589814 0.91 EGFR (0.94) EGFRMAPK3ALK
SCHEMBL28053865 0.90 EGFR (0.83) EGFRMAPK3ALK
SCHEMBL28053991 0.90 JAK3 (0.73) EGFRMAPK3ALK
Hydrochloric Acid SCHEMBL28053870 0.89 EGFR (0.82) EGFRMAPK3ALK
SCHEMBL15938213 0.89 MAPK3 (1.00) EGFRMAPK3ALK
SCHEMBL28589279 0.88 ALK (0.71) EGFRMAPK3ALK
SCHEMBL16769540 0.88 ALK (1.00) ALK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106905245-B 2, 4-disubstituted pyrimidines 正大天晴药业集团股份有限公司 2021-06-25 CN disclosed