SCHEMBL2858467

SCHEMBL2858467

O=C(O)c1ccc2c(c1)C(NCc1ccc(C#Cc3ccc(F)cc3)cc1)CCC2

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SSTR3 P32745 5/20 0.48
KDM4E B2RXH2 3/20 0.46
ALDH1A1 P00352 2/20 0.45
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
BACE1 P56817 4/20 0.40
CTSD P07339 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
DHODH Q02127 1/20 0.40
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
TAS1R2 Q8TE23 1/20 0.39
LMNA P02545 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2855184 0.89 KDM4E (0.46) SSTR3KDM4EALDH1A1HDAC1HDAC6
SCHEMBL2857395 0.86 KDM4E (0.48) KDM4EALDH1A1HDAC1HDAC6BACE1
SCHEMBL13711749 0.80 KDM4E (0.48) SSTR3KDM4EALDH1A1HDAC1HDAC6
SCHEMBL5598540 0.79 KDM4E (0.41) SSTR3KDM4EALDH1A1HDAC1HDAC6
SCHEMBL2853430 0.77 TAOK1 (0.48) KDM4EALDH1A1BACE1CTSD
SCHEMBL2853647 0.72 NSD2 (0.38) SSTR3MEN1KMT2A
SCHEMBL785333 0.70 KMT2A (0.49) SSTR3KDM4EMEN1KMT2ADHODH
SCHEMBL785332 0.70 KMT2A (0.49) SSTR3KDM4EMEN1KMT2ADHODH
SCHEMBL13945234 0.70 KDM4E (0.47) SSTR3KDM4EALDH1A1
SCHEMBL18023358 0.70 HDAC1 (0.51) SSTR3ALDH1A1HDAC1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654247-B1 ALKYNYL ARYL CARBOXAMIDES MERCK SERONO SA (CH) 2010-01-20 EP claimed