SCHEMBL28587713

SCHEMBL28587713

CN(C)c1c(C(=O)O)sc2ccccc12.[LiH]

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCL1 Q07820 5/20 0.56
PRNP P04156 1/20 0.48
RXFP1 Q9HBX9 1/20 0.48
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
EDNRA P25101 1/20 0.44
LIMK1 P53667 2/20 0.44
IKBKB O14920 1/20 0.44
CD274 Q9NZQ7 1/20 0.43
KDM4E B2RXH2 1/20 0.43
MEN1 O00255 1/20 0.43
ALDH1A1 P00352 1/20 0.43
GLA P06280 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
HPGD P15428 1/20 0.43
ALOX15 P16050 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17973604 0.98 MCL1 (0.57) MCL1PRNPRXFP1HDAC1HDAC8
SCHEMBL6598312 0.86 MAOB (0.46) MCL1PRNPRXFP1HDAC1HDAC8
Lithium Ion SCHEMBL17960200 0.82 RXFP1 (0.43) MCL1PRNPRXFP1HDAC1HDAC8
SCHEMBL17960110 0.81 LMNA (0.65) RXFP1HDAC1HDAC8HDAC6LMNA
SCHEMBL21874448 0.78 GPR35 (0.45) MCL1PRNPEDNRAPTPN2PTPN1
SCHEMBL17173227 0.78 MCL1 (0.51) MCL1PRNPRXFP1LMNAKDM4E
SCHEMBL584871 0.75 RXFP1 (0.71) MCL1PRNPRXFP1HDAC1HDAC8
SCHEMBL29939764 0.75 RXFP1 (0.71) MCL1PRNPRXFP1HDAC1HDAC8
SCHEMBL346530 0.75 MCL1 (0.62) MCL1PRNPRXFP1HDAC1HDAC8
SCHEMBL28865810 0.75 MCL1 (0.47) MCL1PRNPRXFP1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107873023-B 3-alkyl-4-amido-bicyclo [4, 5, 0] hydroxamic acids as HDAC inhibitors 福马治疗股份有限公司 2021-07-23 CN disclosed