SCHEMBL28588702

SCHEMBL28588702

N#Cc1cccc(COc2ccc(-c3nccc(C(=O)O)n3)cc2)c1Br

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
XDH P47989 11/20 0.54
FFAR1 O14842 2/20 0.43
ALKBH1 Q13686 1/20 0.42
CYP4F2 P78329 1/20 0.41
CYP4A11 Q02928 1/20 0.41
ADAMTS4 O75173 1/20 0.39
MMP13 P45452 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
AKR1B1 P15121 1/20 0.38
MCL1 Q07820 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28583441 0.88 XDH (0.71) XDHFFAR1ALKBH1CYP4F2CYP4A11
SCHEMBL28574824 0.88 XDH (0.54) XDHFFAR1ALKBH1CYP4F2CYP4A11
SCHEMBL28588699 0.88 XDH (0.54) XDHFFAR1ALKBH1CYP4F2CYP4A11
SCHEMBL28587001 0.81 XDH (0.56) XDHFFAR1ALKBH1ADAMTS4MMP13
SCHEMBL28588707 0.80 XDH (0.63) XDHFFAR1CYP4F2CYP4A11MRGPRX4
SCHEMBL28583439 0.78 XDH (0.61) XDHFFAR1ALKBH1CYP4F2CYP4A11
SCHEMBL28568631 0.76 XDH (0.63) XDHCYP4F2CYP4A11MRGPRX4MCL1
SCHEMBL28572338 0.76 XDH (0.63) XDHCYP4F2CYP4A11MRGPRX4MCL1
SCHEMBL28582833 0.76 XDH (0.63) XDHCYP4F2CYP4A11MRGPRX4MCL1
SCHEMBL28574650 0.72 XDH (0.52) XDHCYP4F2CYP4A11MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112979559-A 2-phenyl pyrimidine formic acid derivative and preparation method and application thereof 沈阳药科大学 2021-06-18 CN claimed
CN-112979559-A 2-phenyl pyrimidine formic acid derivative and preparation method and application thereof 沈阳药科大学 2021-06-18 CN disclosed