SCHEMBL28599093

SCHEMBL28599093

NNC(=O)Nc1cc(Cl)cc(Cl)c1.O=C1CC(c2ccc(Br)cc2)Nc2ccc(Cl)cc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LIG1 P18858 1/20 0.39
GRIK1 P39086 1/20 0.36
P2RY1 P47900 1/20 0.34
CNR1 P21554 2/20 0.34
MAPT P10636 3/20 0.34
KDR P35968 2/20 0.34
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
FPR1 P21462 1/20 0.34
FPR2 P25090 1/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 1/20 0.34
POLB P06746 1/20 0.34
GAA P10253 1/20 0.34
NTSR1 P30989 1/20 0.34
HTT P42858 1/20 0.34
P2RX1 P51575 1/20 0.33
P2RX4 Q99571 1/20 0.33
P2RX7 Q99572 1/20 0.33
TMPRSS4 Q9NRS4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28606032 0.95 GRIK1 (0.41) LIG1GRIK1CNR1KDRMEN1
SCHEMBL28614923 0.94 GRIK1 (0.40) LIG1GRIK1CNR1KDRMEN1
SCHEMBL28599139 0.94 GRIK1 (0.40) LIG1GRIK1CNR1KDRMEN1
SCHEMBL28606070 0.91 GRIK1 (0.42) LIG1GRIK1CNR1MAPTKDR
SCHEMBL28598858 0.90 IDH1 (0.38) LIG1GRIK1CNR1MAPTKDR
SCHEMBL28598799 0.90 IDH1 (0.38) LIG1GRIK1CNR1MAPTKDR
SCHEMBL28608487 0.90 ALDH1A1 (0.38) P2RY1MAPTKDRMEN1KMT2A
SCHEMBL28606031 0.90 MAPT (0.40) MAPTMEN1KMT2AKDM4EALDH1A1
SCHEMBL28608062 0.88 GRIK1 (0.40) LIG1GRIK1CNR1KDRALDH1A1
SCHEMBL28599108 0.88 FPR1 (0.47) GRIK1MEN1KMT2AFPR1FPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108558756-B 2-aryl-2, 3-dihydro-4 (1H) -quinolinone semicarbazone compound and application thereof 沈阳药科大学 2021-08-03 CN claimed