SCHEMBL28599137

SCHEMBL28599137

NNC(=O)Nc1ccc(Br)cc1.O=C1CC(c2ccc(Cl)cc2Cl)Nc2ccccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.40
KDM4E B2RXH2 2/20 0.40
HTT P42858 2/20 0.40
CYP1A2 P05177 1/20 0.40
GAA P10253 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
ALOX12 P18054 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDR P35968 4/20 0.39
MAPT P10636 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
CASP3 P42574 1/20 0.38
RAB9A P51151 1/20 0.38
SENP8 Q96LD8 1/20 0.38
SENP7 Q9BQF6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28600917 0.93 GRIK1 (0.39) LMNAKDRMAPTMEN1KMT2A
SCHEMBL28601601 0.91 ALDH1A1 (0.42) LMNAKDM4EHTTCYP1A2GAA
SCHEMBL28612436 0.90 HTT (0.42) LMNAKDM4EHTTCYP1A2GAA
SCHEMBL28612707 0.88 MEN1 (0.41) KDM4EHTTCYP2C9CYP2C19SMN1; SMN2
SCHEMBL28606352 0.88 AR (0.42) LMNAKDM4EHTTCYP1A2GAA
SCHEMBL28618559 0.88 MEN1 (0.41) LMNAKDM4EHTTCYP1A2GAA
SCHEMBL28603909 0.87 KDR (0.40) LMNAKDRMAPTMEN1KMT2A
SCHEMBL28608385 0.87 KDM4E (0.43) LMNAKDM4EHTTCYP1A2GAA
SCHEMBL28614837 0.87 KDR (0.40) LMNAKDRMAPTMEN1KMT2A
SCHEMBL28606070 0.85 GRIK1 (0.42) LMNAKDRMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108558756-B 2-aryl-2, 3-dihydro-4 (1H) -quinolinone semicarbazone compound and application thereof 沈阳药科大学 2021-08-03 CN claimed