SCHEMBL285997

SCHEMBL285997

CCCCc1noc(C)c1C=Cc1nc(C)c(C(=O)OC(C)C(N)=O)s1

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.36
TSHR P16473 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL285901 0.86 POLB (0.42) KMT2ATSHRPOLB
SCHEMBL285902 0.86 POLB (0.42) KMT2ATSHRPOLB
SCHEMBL285868 0.86 IKBKB (0.35)
SCHEMBL285869 0.86 IKBKB (0.35)
SCHEMBL285784 0.85 TSHR (0.35) KMT2ATSHRPOLB
SCHEMBL285699 0.83 GABRA5 (0.43) POLB
SCHEMBL285701 0.83 GABRA5 (0.43) POLB
SCHEMBL286202 0.82 ALDH1A1 (0.38) TSHR
SCHEMBL2749746 0.82 ALDH1A1 (0.38) TSHR
SCHEMBL286203 0.82 ALDH1A1 (0.38) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2427459-A1 ISOXAZOLE-THIAZOLE DERIVATIVES AS GABA A RECEPTOR INVERSE AGONISTS FOR USE IN THE TREATMENT OF COGNITIVE DISORDERS F. Hoffmann-La Roche AG (CH) 2012-03-14 EP disclosed