SCHEMBL28600101

SCHEMBL28600101

CCOCCOc1ccc(-c2cc(N)nc(N)n2)cc1

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.60
NCF1 P14598 6/20 0.53
MAOB P27338 5/20 0.50
MAOA P21397 3/20 0.50
ACHE P22303 2/20 0.50
XDH P47989 1/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46
HRH2 P25021 1/20 0.45
HRH3 Q9Y5N1 1/20 0.45
DHFR P00374 2/20 0.43
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 1/20 0.42
CYP19A1 P11511 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
BCHE P06276 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30488037 1.00 DYRK1A (0.60) DYRK1ANCF1MAOBMAOAACHE
SCHEMBL28589316 0.81 DYRK1A (0.60) DYRK1AMAOBMAOAACHEXDH
SCHEMBL30488024 0.81 DYRK1A (0.60) DYRK1AMAOBMAOAACHEXDH
SCHEMBL30488027 0.81 DYRK1A (0.60) DYRK1AMAOBMAOAACHEXDH
SCHEMBL1388722 0.76 DYRK1A (1.00) DYRK1AMAOBMAOAACHENPC1
SCHEMBL28589976 0.76 ACHE (0.58) DYRK1AMAOBMAOAACHENPC1
SCHEMBL30488017 0.76 ACHE (0.58) DYRK1AMAOBMAOAACHENPC1
SCHEMBL28707075 0.75 CYP2D6 (0.56) NCF1XDHNPC1RAB9AALDH1A1
SCHEMBL4059613 0.75 RARB (0.53) NCF1ALDH1A1CYP1A2CYP2D6CYP19A1
SCHEMBL4061378 0.73 NQO1 (0.57) NCF1ALDH1A1MAPK1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113061116-B Aminopyrimidine compound, preparation method, composition and application thereof 上海医药工业研究院 2023-07-25 CN disclosed
CN-113061116-A Aminopyrimidine compound, preparation method, composition and application thereof 上海医药工业研究院 2021-07-02 CN disclosed