SCHEMBL30488024

SCHEMBL30488024

Nc1cc(-c2ccc(OCCBr)cc2)nc(N)n1

nearest known ligand 0.60

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 3/20 0.60
MAOB P27338 7/20 0.54
MAOA P21397 5/20 0.54
ACHE P22303 2/20 0.54
BCHE P06276 1/20 0.44
XDH P47989 3/20 0.43
HRH2 P25021 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
KDM4E B2RXH2 1/20 0.40
DHFR P00374 2/20 0.40
CYP1A1 P04798 1/20 0.40
CYP1B1 Q16678 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA1 P30542 1/20 0.40
NPC1 O15118 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MAPK1 P28482 1/20 0.39
RAB9A P51151 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30488027 1.00 DYRK1A (0.60) DYRK1AMAOBMAOAACHEBCHE
SCHEMBL28589316 1.00 DYRK1A (0.60) DYRK1AMAOBMAOAACHEBCHE
SCHEMBL28600101 0.81 DYRK1A (0.60) DYRK1AMAOBMAOAACHEBCHE
SCHEMBL30488037 0.81 DYRK1A (0.60) DYRK1AMAOBMAOAACHEBCHE
SCHEMBL30488017 0.76 ACHE (0.58) DYRK1AMAOBMAOAACHEBCHE
SCHEMBL28589976 0.76 ACHE (0.58) DYRK1AMAOBMAOAACHEBCHE
SCHEMBL1388722 0.76 DYRK1A (1.00) DYRK1AMAOBMAOAACHEHRH2
SCHEMBL28586101 0.72 DYRK1A (0.64) DYRK1AMAOBMAOAACHEHRH2
SCHEMBL30488021 0.72 DYRK1A (0.64) DYRK1AMAOBMAOAACHEHRH2
SCHEMBL29237867 0.72 CYP3A4 (0.47) HRH3NPC1ALDH1A1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113061116-B Aminopyrimidine compound, preparation method, composition and application thereof 上海医药工业研究院 2023-07-25 CN disclosed