SCHEMBL28600318

SCHEMBL28600318

Cc1cc(Br)cc2c1C(=O)N(C)CC2

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
GRM5 P41594 1/20 0.35
BRD4 O60885 3/20 0.34
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
NPSR1 Q6W5P4 1/20 0.33
SRD5A1 P18405 1/20 0.33
HTR2A P28223 1/20 0.31
HTR2C P28335 1/20 0.31
HTR2B P41595 1/20 0.31
MAPT P10636 1/20 0.31
DRD2 P14416 1/20 0.31
TNKS O95271 1/20 0.31
PARP1 P09874 1/20 0.31
TNKS2 Q9H2K2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29209082 0.83 BRD4 (0.42) MEN1KMT2ABRD4HTR2AHTR2C
SCHEMBL13139310 0.83 HTR2A (0.44) MEN1KMT2AGRM5BRD4GAA
SCHEMBL28597676 0.80 MEN1 (0.55) MEN1KMT2AGRM5BRD4GAA
SCHEMBL8749812 0.73 TAS1R3 (0.32) SRD5A1
SCHEMBL25256410 0.73 MEN1 (0.41) MEN1KMT2AGRM5BRD4GAA
SCHEMBL24771273 0.73 SRD5A1 (0.36) BRD4NPSR1SRD5A1
SCHEMBL30723049 0.73 SRD5A1 (0.36) BRD4NPSR1SRD5A1
SCHEMBL12715961 0.72 HTR2A (0.44) MEN1KMT2AGRM5HTR2AHTR2C
SCHEMBL4751133 0.71 TAS1R3 (0.34) BRD4HTR2AHTR2CHTR2BMAPT
SCHEMBL172065 0.71 GRM5 (0.56) MEN1KMT2AGRM5BRD4SRD5A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113166139-A Pyrrolo [2,3-b ] pyridines as HPK1 inhibitors and uses thereof 百济神州有限公司 2021-07-23 CN disclosed