SCHEMBL28600366

SCHEMBL28600366

CC(C)(C)OC(=O)Nc1cc(C(F)(F)F)cs1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXFP1 Q9HBX9 1/20 0.43
LMNA P02545 1/20 0.38
POLB P06746 1/20 0.38
CACNA1H O95180 1/20 0.37
CACNA1B Q00975 1/20 0.37
CACNA1C Q13936 1/20 0.37
GPR35 Q9HC97 1/20 0.36
METAP1 P53582 1/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
TRPA1 O75762 1/20 0.35
KCNQ4 P56696 1/20 0.35
KCNQ5 Q9NR82 1/20 0.35
PTPRB P23467 1/20 0.35
CYP17A1 P05093 1/20 0.35
MAPT P10636 2/20 0.34
STS P08842 1/20 0.34
P2RY14 Q15391 1/20 0.34
PTPN5 P54829 1/20 0.34
CA1 P00915 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28834318 0.81 KCNQ4 (0.41) RXFP1LMNAPOLBMETAP1KCNQ4
SCHEMBL437388 0.80 LCK (0.45) CYP17A1CA1CA2
SCHEMBL1352029 0.80 RAF1 (0.48) CYP17A1CA1CA2
SCHEMBL10965342 0.79 MAPT (0.48) GPR35MAPTCA1CA2
SCHEMBL28834313 0.78 GAA (0.39) METAP1CYP17A1CA1CA2
SCHEMBL6640279 0.78 CYP17A1 (0.36) METAP1KCNQ4KCNQ5CYP17A1CA1
SCHEMBL27620314 0.77 MAPT (0.43) METAP1CYP17A1MAPTCA1CA2
SCHEMBL438824 0.76 CYP17A1 (0.35) METAP1KCNQ4KCNQ5CYP17A1CA1
SCHEMBL25360784 0.75 EGLN2 (0.41) TRPA1KCNQ4KCNQ5CYP17A1CA1
SCHEMBL8574413 0.74 MAPT (0.57) RXFP1LMNAGPR35TRPA1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112939829-B Synthetic method of aryl trifluoromethyl thioether 武汉药明康德新药开发有限公司 2023-02-21 CN disclosed
CN-112939829-A Synthetic method of aryl trifluoromethyl thioether 武汉药明康德新药开发有限公司 2021-06-11 CN disclosed