SCHEMBL28601037

SCHEMBL28601037

Cc1cccn2c(NC(C)(C)C)c(-c3ccco3)nc12

nearest known ligand 0.70

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
GAA P10253 14/20 0.70
SMN1; SMN2 Q16637 6/20 0.70
TP53 P04637 4/20 0.70
HPGD P15428 4/20 0.45
MAPT P10636 9/20 0.43
BRD4 O60885 1/20 0.43
ALDH1A1 P00352 4/20 0.43
HTT P42858 3/20 0.43
KDM4E B2RXH2 2/20 0.43
TDP1 Q9NUW8 1/20 0.41
ADRA1B P35368 1/20 0.40
LMNA P02545 1/20 0.40
POLB P06746 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
HSD17B10 Q99714 1/20 0.40
PKM P14618 1/20 0.40
NPY1R P25929 1/20 0.40
NPY2R P49146 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20889799 0.80 GAA (0.67) GAASMN1; SMN2TP53HPGDMAPT
SCHEMBL6649705 0.79 ADRA1B (0.64) GAASMN1; SMN2TP53HPGDMAPT
SCHEMBL5167267 0.78 ALOX5 (0.65) GAASMN1; SMN2TP53HPGDMAPT
SCHEMBL6650196 0.77 GAA (0.61) GAASMN1; SMN2TP53HPGDMAPT
SCHEMBL28599553 0.76 MAPT (0.56) GAASMN1; SMN2TP53HPGDMAPT
SCHEMBL6652519 0.75 GAA (0.72) GAASMN1; SMN2TP53HPGDMAPT
SCHEMBL4717242 0.75 IDO1 (0.65) GAASMN1; SMN2TP53HPGDMAPT
SCHEMBL20889821 0.74 SALL4 (0.55) GAASMN1; SMN2TP53HPGDMAPT
SCHEMBL17833795 0.72 BRD4 (0.78) GAAMAPTBRD4
SCHEMBL28609935 0.71 GAA (0.68) GAASMN1; SMN2TP53HPGDMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109096139-B Preparation method of alpha-carbonyl amide derivative 贵州大学 2021-03-02 CN disclosed