SCHEMBL28601435

SCHEMBL28601435

Cc1nc(C)c(C(=O)NCCc2c[nH]c3ccccc23)nc1C

nearest known ligand 0.67

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 5/20 0.67
NPC1 O15118 5/20 0.64
RAB9A P51151 5/20 0.64
MEN1 O00255 3/20 0.64
KMT2A Q03164 3/20 0.64
LMNA P02545 1/20 0.63
CYP1A2 P05177 1/20 0.63
PKM P14618 1/20 0.63
TSHR P16473 1/20 0.63
CYP2C19 P33261 1/20 0.63
BLM P54132 1/20 0.63
CDK4 P11802 2/20 0.61
CCND1 P24385 2/20 0.61
PTGS2 P35354 3/20 0.60
PTGS1 P23219 2/20 0.60
ATM Q13315 1/20 0.60
POLB P06746 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28602534 0.80 CA12 (0.56) SIRT1MEN1KMT2A
SCHEMBL6394942 0.79 MEN1 (0.76) SIRT1NPC1RAB9AMEN1KMT2A
SCHEMBL28045701 0.79 NPC1 (0.78) SIRT1NPC1RAB9AMEN1KMT2A
SCHEMBL4331421 0.78 MEN1 (1.00) SIRT1NPC1RAB9AMEN1KMT2A
Nb-Acetyltryptamine SCHEMBL468850 0.78 MEN1 (1.00) SIRT1NPC1RAB9AMEN1KMT2A
SCHEMBL15145374 0.77 PTGS1 (0.75) SIRT1NPC1RAB9AMEN1KMT2A
Nb-Acetyltryptamine SCHEMBL29669230 0.77 MEN1 (0.97) SIRT1NPC1RAB9AMEN1KMT2A
SCHEMBL28477305 0.76 PTGS1 (0.78) SIRT1NPC1RAB9AMEN1KMT2A
SCHEMBL14198238 0.76 CDK4 (0.77) SIRT1NPC1RAB9AMEN1KMT2A
SCHEMBL15145387 0.76 SIRT1 (0.76) SIRT1NPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112961143-A Ligustrazine derivative and preparation method thereof 河南省人民医院 2021-06-15 CN claimed