SCHEMBL28601559

SCHEMBL28601559

CC(C)(C)NC(=O)O[C@@H]1CCCN(c2ncc(C(F)(F)F)cc2Br)C1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACACB O00763 2/20 0.43
SMN1; SMN2 Q16637 4/20 0.42
MEN1 O00255 3/20 0.42
KMT2A Q03164 3/20 0.42
LMNA P02545 3/20 0.42
ALDH1A1 P00352 2/20 0.42
CYP2C9 P11712 3/20 0.41
CYP2C19 P33261 3/20 0.41
KDM4E B2RXH2 3/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
SCN10A Q9Y5Y9 4/20 0.41
HPGD P15428 1/20 0.40
PTGS1 P23219 1/20 0.40
PTGS2 P35354 1/20 0.40
HRH3 Q9Y5N1 1/20 0.40
POLB P06746 2/20 0.39
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28614149 0.90 MEN1 (0.43) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28605624 0.89 SMN1; SMN2 (0.53) SMN1; SMN2MEN1KMT2ALMNAALDH1A1
SCHEMBL28614142 0.89 SMN1; SMN2 (0.53) SMN1; SMN2MEN1KMT2ALMNAALDH1A1
SCHEMBL28597276 0.89 ACACB (0.51) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28593886 0.85 ACACB (0.57) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28607800 0.85 CYP2C9 (0.45) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28607796 0.85 CYP2C9 (0.45) ACACBSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL28610083 0.82 MEN1 (0.38) SMN1; SMN2MEN1KMT2ALMNAALDH1A1
SCHEMBL31124462 0.79 SYK (0.51) MEN1KMT2A
SCHEMBL28601560 0.79 SYK (0.51) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113164461-A Heterocyclic derivatives as Nav1.7 and Nav1.8 blockers 拉夸里亚创药株式会社 2021-07-23 CN disclosed