SCHEMBL28601708

SCHEMBL28601708

FC(F)(F)COc1cnc(Cl)c(Cl)c1

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.44
MAPT P10636 2/20 0.44
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
L3MBTL1 Q9Y468 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
KDM4E B2RXH2 1/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
HSP90AA1 P07900 1/20 0.36
HSP90AB1 P08238 1/20 0.36
THRB P10828 1/20 0.36
G6PD P11413 1/20 0.36
ALOX15 P16050 1/20 0.36
CASP1 P29466 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36
CNR2 P34972 2/20 0.36
EPHX2 P34913 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15918588 0.84 MAPT (0.43) ALDH1A1MAPTL3MBTL1KDM4EMEN1
SCHEMBL16011537 0.82 ALDH1A1 (0.42) ALDH1A1MAPT
SCHEMBL14720949 0.79 CHRNB2 (0.45) CHRNB2CHRNA4
SCHEMBL2305437 0.77 SLC7A5 (0.40) ALDH1A1CHRNB2CHRNA4
SCHEMBL12609890 0.76 MAPT (0.45) ALDH1A1MAPTL3MBTL1TDP1KDM4E
SCHEMBL23677159 0.76 SCN9A (0.41) ALDH1A1MAPTL3MBTL1KDM4EMEN1
SCHEMBL16462088 0.76 MAPT (0.37) ALDH1A1MAPTL3MBTL1KDM4EMEN1
SCHEMBL16711868 0.76 ALDH1A1 (0.44) ALDH1A1MAPTKDM4EMEN1KMT2A
SCHEMBL20910481 0.75 SCN9A (0.40) ALDH1A1MEN1KMT2A
SCHEMBL15918740 0.75 ALDH1A1 (0.50) ALDH1A1CHRNB2CHRNA4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113164461-A Heterocyclic derivatives as Nav1.7 and Nav1.8 blockers 拉夸里亚创药株式会社 2021-07-23 CN disclosed