SCHEMBL2860286

SCHEMBL2860286

Cc1c(C(=O)Nc2ccccc2)cnn1-c1ccccc1

nearest known ligand 0.87

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 17/20 0.87
NPC1 O15118 16/20 0.87
NAMPT P43490 1/20 0.81
PKM P14618 3/20 0.79
HPGD P15428 2/20 0.79
NFKB1 P19838 1/20 0.79
NFKB2 Q00653 1/20 0.79
RELA Q04206 1/20 0.79
SMN1; SMN2 Q16637 1/20 0.79
POLB P06746 1/20 0.73
MAPK1 P28482 1/20 0.70
MEN1 O00255 1/20 0.70
KMT2A Q03164 1/20 0.70
MAPT P10636 1/20 0.70

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2857152 0.88 NPC1 (0.91) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL10367090 0.85 HPGD (0.72) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL31610081 0.84 RAB9A (0.71) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL28704189 0.84 HPGD (0.71) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL2544046 0.83 MAPK1 (1.00) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL14132462 0.82 NPC1 (1.00) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL2854522 0.81 MAPK1 (0.64) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL2605692 0.81 HPGD (0.76) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL27405 0.81 MAPK1 (0.78) RAB9ANPC1NAMPTPKMHPGD
SCHEMBL16615777 0.80 NPC1 (0.66) RAB9ANPC1NAMPTPKMHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP claimed
EP-1451160-B1 PYRAZOLE-AMIDES FOR USE IN THE TREATMENT OF PAIN ICAGEN INC (US) 2010-01-13 EP disclosed