SCHEMBL28604236

SCHEMBL28604236

CCOc1ccc2c([c]cn2C(=O)OC(C)(C)C)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR119 Q8TDV5 2/20 0.40
BRD4 O60885 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
MAPT P10636 4/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 3/20 0.36
MMP13 P45452 1/20 0.36
HTR6 P50406 1/20 0.36
AKR1C3 P42330 1/20 0.36
AKR1C2 P52895 1/20 0.36
LMNA P02545 1/20 0.36
KDM4E B2RXH2 2/20 0.36
GAA P10253 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
MEN1 O00255 1/20 0.36
USP2 O75604 1/20 0.36
TSHR P16473 1/20 0.36
MAPK1 P28482 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28600582 0.86 ALDH1A1 (0.41) GPR119BRD4L3MBTL1MAPTALDH1A1
SCHEMBL1948855 0.76 BCHE (0.44) GPR119L3MBTL1ALDH1A1KDM4EMEN1
SCHEMBL28600580 0.75 ALDH1A1 (0.41) GPR119BRD4MAPTALDH1A1LMNA
SCHEMBL2879064 0.74 MCL1 (0.42) GPR119BRD4L3MBTL1MAPTALDH1A1
SCHEMBL31370509 0.74 L3MBTL1 (0.49) GPR119BRD4L3MBTL1MAPTALDH1A1
SCHEMBL17690275 0.70 NR1H2 (0.45) GPR119BRD4MAPTALDH1A1HPGD
SCHEMBL3892320 0.68 ESR2 (0.56) GPR119L3MBTL1MAPTALDH1A1HPGD
SCHEMBL5952979 0.68 MAPT (0.39) GPR119BRD4L3MBTL1MAPTALDH1A1
SCHEMBL25736835 0.68 MAPT (0.46) GPR119BRD4L3MBTL1MAPTALDH1A1
SCHEMBL14051459 0.68 L3MBTL1 (0.46) GPR119L3MBTL1HTR6AKR1C3NR1H2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113105459-A Triazolopyrimidine derivative and preparation method and application thereof 五邑大学 2021-07-13 CN claimed
CN-113105459-B Triazolopyrimidine derivative and preparation method and application thereof 五邑大学 2022-05-03 CN disclosed
CN-113105459-A Triazolopyrimidine derivative and preparation method and application thereof 五邑大学 2021-07-13 CN disclosed