SCHEMBL28604348

SCHEMBL28604348

COC(=O)C1CN(C(=O)c2cc(OCc3ccccc3)c(OCc3ccccc3)c(OCc3ccccc3)c2)CCN1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GLRA1 P23415 1/20 0.47
HSD17B10 Q99714 1/20 0.43
ALDH1A1 P00352 4/20 0.43
HPGD P15428 3/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TSHR P16473 1/20 0.42
LMNA P02545 2/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CSF1R P07333 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
PARP1 P09874 1/20 0.41
CYP1A2 P05177 1/20 0.40
SMPD1 P17405 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7656754 0.81 SIGMAR1 (0.51) ALDH1A1HPGDMEN1KMT2ALMNA
SCHEMBL28406248 0.80 PARP1 (0.59) GLRA1HSD17B10ALDH1A1HPGDTSHR
SCHEMBL9781914 0.79 PKM (0.54) ALDH1A1KMT2ACYP1A2
SCHEMBL28919582 0.79 NR1H2 (0.45) GLRA1HSD17B10ALDH1A1HPGDMEN1
SCHEMBL12324603 0.78 SMN1; SMN2 (0.52) MEN1KMT2ASMN1; SMN2NPSR1NPC1
SCHEMBL14646669 0.78 SMN1; SMN2 (0.52) MEN1KMT2ASMN1; SMN2NPSR1NPC1
SCHEMBL2680992 0.78 SMN1; SMN2 (0.52) MEN1KMT2ASMN1; SMN2NPSR1NPC1
Hydrochloric Acid SCHEMBL29121517 0.77 SMN1; SMN2 (0.51) MEN1KMT2ATSHRSMN1; SMN2NPSR1
SCHEMBL28599521 0.77 SMN1; SMN2 (0.41) GLRA1HSD17B10HPGDLMNASMN1; SMN2
SCHEMBL28236192 0.76 GLRA1 (0.51) GLRA1HSD17B10ALDH1A1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113105395-B 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2022-06-17 CN disclosed
CN-113105395-A 4-phenylsulfonyl-1-trihydroxy benzoyl piperazine-2-carboxamide derivative and preparation method and application thereof 山东大学 2021-07-13 CN disclosed