SCHEMBL28604692

SCHEMBL28604692

N#Cc1cn(Cc2ccccc2)c2ccc(-c3nnn[nH]3)cc12

nearest known ligand 0.64

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.55
ALDH1A1 P00352 2/20 0.55
KMT2A Q03164 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
TDP1 Q9NUW8 2/20 0.55
TSHR P16473 1/20 0.55
KDM4E B2RXH2 1/20 0.48
HTT P42858 1/20 0.48
HSD17B10 Q99714 1/20 0.48
XDH P47989 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28587916 0.90 XDH (0.48) MEN1ALDH1A1KMT2ASMN1; SMN2TDP1
SCHEMBL28591848 0.89 XDH (0.48) XDH
SCHEMBL28604694 0.89 MEN1 (0.42) MEN1ALDH1A1KMT2ASMN1; SMN2TDP1
SCHEMBL28609476 0.89 XDH (0.48) MEN1ALDH1A1KMT2ASMN1; SMN2TDP1
SCHEMBL28591847 0.87 XDH (0.50) XDH
SCHEMBL28592166 0.85 ALDH1A1 (0.45) ALDH1A1SMN1; SMN2XDH
SCHEMBL28594483 0.83 MAPT (0.42) ALDH1A1SMN1; SMN2TSHRHTTXDH
SCHEMBL28596769 0.82 XDH (0.49) XDH
SCHEMBL28609035 0.82 XDH (0.44) ALDH1A1KDM4EXDH
SCHEMBL28613223 0.81 XDH (0.63) XDH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113173917-B 1-alkyl-5-tetrazolyl/pyrimidone-1H-indole-3-carbonitrile compound and preparation method and application thereof 沈阳药科大学 2022-04-08 CN claimed
CN-113173917-A 1-alkyl-5-tetrazolyl/pyrimidone-1H-indole-3-carbonitrile compound and preparation method and application thereof 沈阳药科大学 2021-07-27 CN claimed
CN-113173917-B 1-alkyl-5-tetrazolyl/pyrimidone-1H-indole-3-carbonitrile compound and preparation method and application thereof 沈阳药科大学 2022-04-08 CN disclosed
CN-113173917-A 1-alkyl-5-tetrazolyl/pyrimidone-1H-indole-3-carbonitrile compound and preparation method and application thereof 沈阳药科大学 2021-07-27 CN disclosed