SCHEMBL28607828

SCHEMBL28607828

Cc1cccc(C(=O)NCC2CCOCC2)c1C

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 5/20 0.52
NPC1 O15118 2/20 0.52
RAB9A P51151 1/20 0.52
CNR2 P34972 10/20 0.49
CNR1 P21554 2/20 0.47
TAS1R3 Q7RTX0 1/20 0.47
TAS1R1 Q7RTX1 1/20 0.47
TAS1R2 Q8TE23 1/20 0.47
HTR4 Q13639 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28503120 0.92 P2RX7 (0.47) P2RX7NPC1RAB9ACNR2TAS1R3
SCHEMBL13162628 0.89 NPC1 (0.51) P2RX7NPC1RAB9ACNR2CNR1
SCHEMBL28602013 0.84 CHRM1 (0.60) HTR4
SCHEMBL13161996 0.81 NAMPT (0.50) P2RX7NPC1RAB9A
SCHEMBL20477095 0.79 SMN1; SMN2 (0.57) P2RX7NPC1RAB9ACNR2TAS1R3
SCHEMBL12476380 0.78 CNR1 (0.71) NPC1CNR2CNR1
SCHEMBL8297083 0.78 HPGD (0.57) P2RX7NPC1RAB9A
SCHEMBL28729042 0.78 CNR2 (0.49) NPC1RAB9ACNR2CNR1HTR4
SCHEMBL12697364 0.76 CNR2 (0.56) CNR2CNR1
SCHEMBL13163160 0.76 MEN1 (0.51) P2RX7NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113195497-A Novel imidazopyrazine derivatives 豪夫迈·罗氏有限公司 2021-07-30 CN claimed
CN-113195497-A Novel imidazopyrazine derivatives 豪夫迈·罗氏有限公司 2021-07-30 CN disclosed