SCHEMBL28602013

SCHEMBL28602013

Cc1cccc(C(=O)NCC2CCNCC2)c1C

nearest known ligand 0.60

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 16/20 0.60
CHRM2 P08172 3/20 0.58
CHRM4 P08173 3/20 0.58
CHRM3 P20309 3/20 0.58
CHRM5 P08912 2/20 0.58
HTR4 Q13639 4/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13162900 0.89 CHRM1 (0.65) CHRM1CHRM2CHRM4CHRM3CHRM5
SCHEMBL28600527 0.87 CHRM1 (0.57) CHRM1CHRM2CHRM4CHRM3CHRM5
Hydrochloric Acid SCHEMBL28982241 0.86 CHRM1 (0.56) CHRM1CHRM2CHRM4CHRM3CHRM5
SCHEMBL28607828 0.84 P2RX7 (0.52) HTR4
SCHEMBL22122848 0.80 CHRM1 (0.58) CHRM1CHRM2CHRM4CHRM3CHRM5
SCHEMBL28503120 0.79 P2RX7 (0.47)
SCHEMBL22123764 0.79 TAS1R3 (0.57) HTR4
SCHEMBL13543095 0.78 CHRM1 (0.62) CHRM1CHRM2CHRM4CHRM3CHRM5
SCHEMBL8297083 0.78 HPGD (0.57) CHRM1CHRM2CHRM4CHRM3CHRM5
SCHEMBL7213953 0.77 HTR4 (0.61) CHRM1CHRM2CHRM4CHRM3CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113195497-A Novel imidazopyrazine derivatives 豪夫迈·罗氏有限公司 2021-07-30 CN claimed
CN-113195497-A Novel imidazopyrazine derivatives 豪夫迈·罗氏有限公司 2021-07-30 CN disclosed