SCHEMBL28608304

SCHEMBL28608304

COC(=O)CCC=CCC(NC(=O)OC(C)(C)C)C(=O)OC

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CTSK P43235 11/20 0.48
CYP1A2 P05177 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HTT P42858 1/20 0.40
CTSS P25774 8/20 0.40
NFKB1 P19838 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
CTSL P07711 1/20 0.39
CTSB P07858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
CAPN1 P07384 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
KLK5 Q9Y337 1/20 0.36
CYP2D6 P10635 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16330414 0.89 CTSK (0.54) CTSKCYP1A2CYP2C9CYP2C19HTT
SCHEMBL17884307 0.89 CTSK (0.54) CTSKCYP1A2CYP2C9CYP2C19HTT
SCHEMBL17880452 0.83 CTSK (0.49) CTSKCYP1A2CYP2C9CYP2C19HTT
SCHEMBL17880416 0.83 CTSK (0.49) CTSKCYP1A2CYP2C9CYP2C19HTT
SCHEMBL16330411 0.82 CTSK (0.48) CTSKCYP1A2CYP2C9CYP2C19HTT
SCHEMBL17189629 0.81 AKT1 (0.37) NFKB1SMN1; SMN2CA1CA2CA7
SCHEMBL1317487 0.80 CYP1A2 (0.49) CTSKCYP1A2CYP2C9CYP2C19HTT
SCHEMBL1763873 0.80 CYP1A2 (0.49) CTSKCYP1A2CYP2C9CYP2C19HTT
SCHEMBL2225458 0.80 CYP1A2 (0.49) CTSKCYP1A2CYP2C9CYP2C19HTT
SCHEMBL17884342 0.80 CTSK (0.44) CTSKCYP1A2CYP2C9CYP2C19HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113195473-B Tricyclic compound as STING agonist and preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2022-11-22 CN disclosed
CN-113195473-A Tricyclic compound as STING agonist and preparation method and medical application thereof 江苏恒瑞医药股份有限公司 2021-07-30 CN disclosed