SCHEMBL28609236

SCHEMBL28609236

O=C(Nc1cc2c(s1)CCC(NC(=O)C(F)(F)F)C2)C1CC1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.36
ALOX15 P16050 1/20 0.36
NPC1 O15118 7/20 0.34
RAB9A P51151 7/20 0.34
MTNR1A P48039 3/20 0.33
MTNR1B P49286 3/20 0.33
ALDH1A1 P00352 3/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
RAF1 P04049 2/20 0.31
BRAF P15056 2/20 0.31
GAA P10253 1/20 0.31
PRNP P04156 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28622749 1.00 TP53 (0.36) TP53ALOX15NPC1RAB9AMTNR1A
SCHEMBL27415382 0.88 ABL1 (0.34) NPC1RAB9AALDH1A1
SCHEMBL27415416 0.87 NPC1 (0.32) NPC1RAB9AALDH1A1
SCHEMBL21597854 0.85 TP53 (0.41) TP53ALOX15NPC1RAB9AMTNR1A
SCHEMBL21603867 0.82 TP53 (0.39) TP53ALOX15NPC1RAB9AMTNR1A
SCHEMBL21603763 0.78 TP53 (0.39) TP53ALOX15NPC1RAB9AALDH1A1
SCHEMBL21597801 0.76 TP53 (0.40) TP53ALOX15NPC1RAB9AALDH1A1
SCHEMBL21597427 0.76 TBXAS1 (0.46) TP53ALOX15NPC1RAB9AALDH1A1
SCHEMBL21603764 0.76 ALDH1A1 (0.54) TP53ALOX15NPC1RAB9AALDH1A1
SCHEMBL21603808 0.75 EPHX2 (0.50) NPC1RAB9AMTNR1AMTNR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-112566910-A Thiophene derivatives for the treatment of IgE induced diseases UCB生物制药有限责任公司 2021-03-26 CN disclosed