Bicarbonate

Bicarbonate

SCHEMBL28609581

Clc1cnccc1Br.N.O=C(O)O.O=C(O)O

nearest known ligand 0.42

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

GSK3AGSK3BIMPA1

The experimentally established mechanism targets of Bicarbonate. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.42
CCNC P24863 2/20 0.39
CDK8 P49336 2/20 0.39
ROCK2 O75116 1/20 0.39
ROCK1 Q13464 1/20 0.39
LMNA P02545 2/20 0.38
KMT2A Q03164 5/20 0.37
MEN1 O00255 4/20 0.37
ALDH1A1 P00352 2/20 0.37
KDM4C Q9H3R0 2/20 0.37
MAPT P10636 2/20 0.37
KDM4E B2RXH2 2/20 0.37
KDM6B O15054 1/20 0.37
KDM4A O75164 1/20 0.37
THRB P10828 1/20 0.37
KDM4D Q6B0I6 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL505164 0.87
SCHEMBL29514226 0.87
Bicarbonate SCHEMBL28392515 0.73 LMNA (0.58) GAAROCK2ROCK1LMNAKMT2A
SCHEMBL116912 0.71 KDM4C (0.59) GAAROCK2ROCK1LMNAKMT2A
SCHEMBL933359 0.71 KDM4C (0.53) GAACCNCCDK8KMT2AMEN1
SCHEMBL30933589 0.71 KDM4C (0.59) GAAROCK2ROCK1LMNAKMT2A
SCHEMBL7431923 0.69 TDP1 (0.41) GAACCNCCDK8ROCK2ROCK1
Hydrochloric Acid SCHEMBL1027775 0.69 KDM4C (0.57) GAAROCK2ROCK1LMNAKMT2A
SCHEMBL360577 0.69
SCHEMBL29571714 0.69

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113149996-B Polycyclic amide derivative as CDK9 inhibitor, and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2022-12-20 CN disclosed
CN-115340555-A Pyridine acetamide derivative as CDK inhibitor, and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2022-11-15 CN disclosed
CN-113173924-B Pyridine acetamide derivative as CDK inhibitor, and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2022-07-19 CN disclosed
CN-113173924-A Pyridine acetamide derivative as CDK inhibitor, and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2021-07-27 CN disclosed
CN-113149996-A Polycyclic amide derivative serving as CDK9 inhibitor, and preparation method and application thereof 苏州阿尔脉生物科技有限公司 2021-07-23 CN disclosed